Aachen papers per year
Papers 18
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Medicinal chemistry of P2 and adenosine receptors: Common scaffolds adapted for multiple targets2020 Biochemical Pharmacology article Biochemistry, Genetics and Molecular Biology Adenosine and Purinergic Signaling Open access cited by 4 patents
Kenneth A. Jacobson, Adriaan P. IJzerman, Christa Elisabeth Müller
45citations -
Integration of temporal single cell cellular stress response activity with logic-ODE modeling reveals activation of ATF4-CHOP axis as a critical predictor of drug-induced liver injury2021 Biochemical Pharmacology article Pharmacology, Toxicology and Pharmaceutics Drug-Induced Hepatotoxicity and Protection Open access
Lukas S. Wijaya, Panuwat Trairatphisan, Attila Gábor, Marije Niemeijer, Jason Keet, Ariadna Alcalà Morera, +13 more
27citations -
Design and pharmacological profile of a novel covalent partial agonist for the adenosine A1 receptor2020 Biochemical Pharmacology article Biochemistry, Genetics and Molecular Biology Adenosine and Purinergic Signaling Open access
Xue Fei Yang, Majlen A. Dilweg, Dion Osemwengie, Lindsey Burggraaff, Daan van der Es, Laura H. Heitman, +1 more
16citations -
G protein-coupled receptors expressed and studied in yeast. The adenosine receptor as a prime example2020 Biochemical Pharmacology article Biochemistry, Genetics and Molecular Biology Receptor Mechanisms and Signaling Open access cited by 1 patent
Xuesong Wang, Gerard J. P. van Westen, Laura H. Heitman, Adriaan P. IJzerman
12citations -
Impact of cancer-associated mutations in CC chemokine receptor 2 on receptor function and antagonism2022 Biochemical Pharmacology article Biochemistry, Genetics and Molecular Biology Receptor Mechanisms and Signaling Open access
Lisa S. den Hollander, Olivier J. M. Béquignon, Xiangzi Wang, K. van Wezel, Jeremy D. Broekhuis, Marina Gorostiola González, +4 more
10citations -
Kinetic profiling and functional characterization of 8-phenylxanthine derivatives as A2B adenosine receptor antagonists2022 Biochemical Pharmacology article Biochemistry, Genetics and Molecular Biology Adenosine and Purinergic Signaling Open access
Anna Vlachodimou, Henk J. de Vries, Milena Pasoli, Miranda Goudswaard, Soon‐Ai Kim, Yong‐Chul Kim, +6 more
9citations -
A kinase inhibitor screen reveals MEK1/2 as a novel therapeutic target to antagonize IGF1R-mediated antiestrogen resistance in ERα-positive luminal breast cancer2022 Biochemical Pharmacology article Biochemistry, Genetics and Molecular Biology Estrogen and related hormone effects Open access
Lynn Wester, Sanne Venneker, M. Hazenoot, Chantal Pont, Esmee Koedoot, John W.M. Martens, +6 more
7citations -
Exploring the binding kinetics of intracellular allosteric antagonists for CC chemokine receptor 2 — a key to improve insurmountable antagonism2026 Biochemical Pharmacology article Biochemistry, Genetics and Molecular Biology Receptor Mechanisms and Signaling Open access
Yao Yao, Lisa S. den Hollander, Bente T.M. Bleijs, Thomas Härtung, Uwe Grether, Natalia V. Ortiz Zacarı́as, +1 more
1citations -
Targeting chitinase-3-like protein-1 in pancolitis by a drug-repurposing approach2026 Biochemical Pharmacology article Biochemistry, Genetics and Molecular Biology Inflammatory Bowel Disease Open access
Faranak Bahramimehr, Stefanie Kurz, Axel Guthart, Susanne M. Krug, Anja Fromm, Damian Tarasek, +11 more
0citations -
Corrigendum to “Impact of cancer-associated mutations in CC chemokine receptor 2 on receptor function and antagonism” [Biochem. Pharmacol. 208 (2023) 115399]
Lisa S. den Hollander, Olivier J. M. Béquignon, Xiangzi Wang, K. van Wezel, Jeremy D. Broekhuis, Marina Gorostiola González, +4 more
0citations -
CC chemokine receptor 2 is allosterically modulated by sodium ions and amiloride derivatives through a distinct sodium ion binding site2024 Biochemical Pharmacology article Biochemistry, Genetics and Molecular Biology Receptor Mechanisms and Signaling
Lisa S. den Hollander, Annelien J.M. Zweemer, Olivier J. M. Béquignon, Dora Hammerl, Bente T.M. Bleijs, Margo Veenhuizen, +5 more
0citations
18 results
Most active Aachen authors
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Laura H. Heitman 7,065 citations overall8 papers
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Adriaan P. IJzerman 28,835 citations overall7 papers
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Gerard J. P. van Westen 6,624 citations overall4 papers
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Lisa S. den Hollander 48 citations overall4 papers
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Olivier J. M. Béquignon 272 citations overall3 papers
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Jeremy D. Broekhuis 47 citations overall3 papers
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Karin E. de Visser 21,572 citations overall2 papers
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Bob van de Water 13,491 citations overall2 papers
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Marina Gorostiola González 634 citations overall2 papers
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Marije Niemeijer 612 citations overall2 papers
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Xiangzi Wang 26 citations overall2 papers
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K. van Wezel 15 citations overall2 papers
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Bente T.M. Bleijs 4 citations overall2 papers
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Julio Sáez-Rodríguez 48,113 citations overall1 paper
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Twan Lammers 36,184 citations overall1 paper