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Deciphering conformational selectivity in the A 2A adenosine G protein-coupled receptor by Free Energy simulations2021 bioRxiv (Cold Spring Harbor Laboratory) preprint Biochemistry, Genetics and Molecular Biology Receptor Mechanisms and Signaling Open access
Willem Jespers, Laura H. Heitman, Adriaan P. IJzerman, Eddy Sotelo, Gerard J. P. van Westen, Johan Åqvist, +1 more
1citations -
Molecular basis of ligand binding and receptor activation at the human A3 adenosine receptor2025 bioRxiv (Cold Spring Harbor Laboratory) preprint Biochemistry, Genetics and Molecular Biology Adenosine and Purinergic Signaling Open access
Liudi Zhang, Jesse I. Mobbs, Felix M. Bennetts, Hariprasad Venugopal, Anh T. N. Nguyen, Arthur Christopoulos, +5 more
1citations -
A universal cannabinoid CB1 and CB2 receptor TR-FRET kinetic ligand binding assay2024 bioRxiv (Cold Spring Harbor Laboratory) preprint Medicine Cannabis and Cannabinoid Research Open access
Leire Borrega Roman, Bradley L. Hoare, Miroslav Kosar, Roman C. Sarott, Kacper J. Patej, Jara Bouma, +15 more
0citations -
Novel assays monitoring direct glucocorticoid receptor protein activity exhibit high predictive power for ligand activity on endogenous gene targets2022 bioRxiv (Cold Spring Harbor Laboratory) preprint Biochemistry, Genetics and Molecular Biology Estrogen and related hormone effects Open access
Laura Van Moortel, Jonathan Thommis, Brecht Maertens, An Staes, Dorien Clarisse, Delphine De Sutter, +5 more
3citations -
Membrane Lipids and Water Shape the Unbinding Kinetics of ZM241385 from Human Adenosine A 2A Receptor Variants2026 bioRxiv (Cold Spring Harbor Laboratory) preprint Biochemistry, Genetics and Molecular Biology Receptor Mechanisms and Signaling Open access
Marta Devodier, Davide Mandelli, Giulia Rossetti, Paolo Carloni
0citations -
Modeling the Orthosteric Binding Site of the G Protein-Coupled Odorant Receptor OR5K12022 bioRxiv (Cold Spring Harbor Laboratory) preprint Biochemistry, Genetics and Molecular Biology Receptor Mechanisms and Signaling Open access
Alessandro Nicoli, Franziska Haag, Patrick Marcinek, Ruiming He, Johanna Kreißl, Jörg Stein, +5 more
2citations -
Selective Serotonin Reuptake Inhibitors Within Cells: Temporal Resolution in Cytoplasm, Endoplasmic Reticulum, and Membrane2022 bioRxiv (Cold Spring Harbor Laboratory) preprint Neuroscience Neuroscience and Neuropharmacology Research Open access
Aaron L. Nichols, Zack Blumenfeld, Laura Luebbert, Hailey J. Knox, Anand K. Muthusamy, Jonathan S. Marvin, +9 more
2citations -
Natural product-derived azaphilones are selective scaffolds for covalent lysine liganding in live cells2026 bioRxiv (Cold Spring Harbor Laboratory) preprint Chemistry Click Chemistry and Applications Open access
Wei Ding, Sophie Brameyer, Susanne H. Kirsch, Birthe Sandargo, Frank Surup, Stephan M. Hacker, +2 more
0citations -
Probing immune signatures of conjugated pattern recognition receptor ligands identifies chimeras with adjuvant and antitumor activity2025 bioRxiv (Cold Spring Harbor Laboratory) preprint Immunology and Microbiology Immunotherapy and Immune Responses Open access
Špela Janež, Samo Guzelj, Marcela Šišić, Ruža Frkanec, Stane Pajk, Lenny Burgmeijer, +2 more
1citations -
A blueprint for high affinity SARS-CoV-2 Mpro inhibitors from activity-based compound library screening guided by analysis of protein dynamics2020 bioRxiv (Cold Spring Harbor Laboratory) preprint Computer Science Computational Drug Discovery Methods Open access
Jonas Goßen, Simone Albani, Anton Hanke, Benjamin Philipp Joseph, Cathrine C. Bergh, Maria Kuzikov, +14 more
5citations -
Parp7 generates an ADP-ribosyl degron that controls negative feedback of androgen signaling2024 bioRxiv (Cold Spring Harbor Laboratory) preprint Medicine Prostate Cancer Treatment and Research Open access
Krzysztof Wierbiłowicz, Chunsong Yang, Ahmed Almaghasilah, Patryk Adam Wesołowski, Philipp Pracht, Natalia M. Dworak, +7 more
0citations -
PROXINAUT: An Automation Platform for Rapid Hit-to-Degrader Discovery2026 bioRxiv (Cold Spring Harbor Laboratory) preprint Biochemistry, Genetics and Molecular Biology Protein Degradation and Inhibitors Open access
Sean M. McKenna, Monika T. Gnatzy, Edith van der Nol, Femke J. Boxman, Chenlu Zhang, Xiaokang Jin, +4 more
0citations