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A 2A Adenosine Receptor Agonists With Last‐Step Enzymatic 18 F‐Labelling Potential (Fluorinase) for Positron Emission Tomography (PET)2025 European Journal of Organic Chemistry article Biochemistry, Genetics and Molecular Biology Adenosine and Purinergic Signaling Open access
Carina Schleidt, Laura H. Heitman, Sergio Dall’Angelo, David O’Hagan, Phillip T. Lowe
0citations -
Cover Feature: Defined Nylon Oligomers Enable Mechanistic Insight Into Enzymatic Polyamide Depolymerization (ChemSusChem 12/2026)2026 ChemSusChem article Biochemistry, Genetics and Molecular Biology Enzyme Catalysis and Immobilization
Sukmanita Dewi, Hendrik Puetz, Ulrich Schwaneberg, Laura Hartmann
0citations -
Electrochemical Impedance Spectroscopy Biosensor Enabling Kinetic Monitoring of Fucosyltransferase Activity2021 ACS Sensors article Biochemistry, Genetics and Molecular Biology Glycosylation and Glycoproteins Research
Viktoria Heine, Tom Kremers, Nora Menzel, Uwe Schnakenberg, Lothar Elling
16citations -
Inhibiting UCH-L5: Rational Design of a Cyclic Ubiquitin-Based Peptide Inhibitor2022 Frontiers in Molecular Biosciences article Biochemistry, Genetics and Molecular Biology Ubiquitin and proteasome pathways Open access
Dharjath S. Hameed, Huib Ovaa, Gerbrand J. van der Heden van Noort, Ayşegül Sapmaz
2citations -
Metagenomics combined with activity-based proteomics point to gut bacterial enzymes that reactivate mycophenolate2022 Gut Microbes article Pharmacology, Toxicology and Pharmaceutics Pharmacogenetics and Drug Metabolism Open access
Joshua B. Simpson, Josh J. Sekela, Amanda L. Graboski, Valentina Borlandelli, Marissa M. Bivins, Natalie K. Barker, +9 more
43citations -
In Silico and Experimental ADAM17 Kinetic Modeling as Basis for Future Screening System for Modulators2022 International Journal of Molecular Sciences article Biochemistry, Genetics and Molecular Biology Protease and Inhibitor Mechanisms Open access cited by 1 patent
Marian Bienstein, Dmitriy Minond, Ulrich Schwaneberg, Mehdi D. Davari, Daniela Yildiz
13citations -
A family of bacterial Josephin-like deubiquitinases with an irreversible cleavage mode2025 Molecular Cell article Biochemistry, Genetics and Molecular Biology Ubiquitin and proteasome pathways Open access
Thomas Hermanns, Susanne Kolek, Matthias Uthoff, Richard A. de Heiden, Monique P. C. Mulder, Ulrich Baumann, +1 more
10citations -
Metagenomics Combined with Activity-Based Proteomics Point to Gut Bacterial Enzymes that Reactivate Mycophenolate2022 medRxiv preprint Pharmacology, Toxicology and Pharmaceutics Pharmacogenetics and Drug Metabolism Open access
Joshua B. Simpson, Josh J. Sekela, Amanda L. Graboski, Valentina Borlandelli, Natalie K. Barker, Alicia A. Sorgen, +8 more
6citations -
A Direct Assay for Measuring the Activity and Inhibition of Coactivator-Associated Arginine Methyltransferase 12022 Biochemistry article Biochemistry, Genetics and Molecular Biology Cancer-related gene regulation Open access
Yurui Zhang, Matthijs J. van Haren, N. Marechal, N. Troffer-Charlier, Vincent Cura, J. Cavarelli, +1 more
3citations -
Modifications of the Prothrombin Active Site S4 Subpocket Confer Resistance to Dabigatran2025 Thrombosis and Haemostasis article Medicine Blood Coagulation and Thrombosis Mechanisms Open access
Viola J.F. Strijbis, Ka Lei Cheung, Dejvid Veizaj, Tessa A. Rutten, Boris Bruin, Pieter H. Reitsma, +2 more
1citations -
Molecular Modeling of Protein–Peptide Complexes Mimicking Factor Xa–Prothrombin Using AlphaFold-Multimer and Molecular Dynamics Simulations for Functional Prediction2026 Journal of Chemical Information and Modeling article Medicine Blood Coagulation and Thrombosis Mechanisms
Dejvid Veizaj, David Alonzo Poole III, Ka Lei Cheung, Jos V. Flier, Pieter H. Reitsma, Daniël Verhoef, +2 more
1citations