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Role of Conserved Tyrosine Lid Residues in the Activation of the M2 Muscarinic Acetylcholine Receptor2023 Molecular Pharmacology article Biochemistry, Genetics and Molecular Biology Receptor Mechanisms and Signaling Open access
Vi Pham, Maria Clazina Cornelia Habben Jansen, Geoff V. Thompson, Laura H. Heitman, Arthur Christopoulos, David M. Thal, +1 more
6citations -
Deciphering the allosteric control of androgen receptor DNA binding by its disordered N-terminal domain2025 Molecular and Cellular Endocrinology article Medicine Prostate Cancer Treatment and Research Open access
Laurens W.H.J. Heling, Adam P. Rofe, Andrea Alegre‐Martí, Vahid Sheikhhassani, Thomas Schmidt, Eva Estébanez‐Perpiñá, +2 more
2citations -
Pilocarpine‐Induced Effects on Salivary Secretion as a Pharmacological Biomarker for Cholinergic Parasympathetic Activation2021 Clinical Pharmacology in Drug Development article Biochemistry, Genetics and Molecular Biology Receptor Mechanisms and Signaling
Nicoline Treijtel, Dorien Groenendaal‐van de Meent, Ingrid N. Michon, Cees Korstanje, John Meijer, Klaus Francke
5citations -
Allosteric control of Ubp6 and the proteasome via a bidirectional switch2022 Nature Communications article Biochemistry, Genetics and Molecular Biology Ubiquitin and proteasome pathways Open access
Ka Ying Sharon Hung, Sven Klumpe, Markus R. Eisele, Suzanne Elsasser, Geng Tian, Shuangwu Sun, +13 more
44citations -
Discovery of isoquinoline sulfonamides as allosteric gyrase inhibitors with activity against fluoroquinolone-resistant bacteria2024 Nature Chemistry article Biochemistry, Genetics and Molecular Biology Cancer therapeutics and mechanisms Open access
Alexander T. Bakker, Ioli Kotsogianni, Mariana Ávalos, Jeroen M. Punt, Bing Liu, Diana Piermarini, +13 more
29citations -
Structure of human spermine oxidase in complex with a highly selective allosteric inhibitor2022 Communications Biology article Biochemistry, Genetics and Molecular Biology Polyamine Metabolism and Applications Open access cited by 1 patent
Elsie Diaz, Suraj Adhikary, Armand W.J.W. Tepper, Daniel Riley, Rodrigo F. Ortiz‐Meoz, Daniel J. Krosky, +12 more
11citations -
Host defence peptide plectasin targets bacterial cell wall precursor lipid II by a calcium-sensitive supramolecular mechanism2024 Nature Microbiology article Immunology and Microbiology Antimicrobial Peptides and Activities Open access
Shehrazade Jekhmane, Maik G. N. Derks, Sourav Maity, Cornelis J. Slingerland, Kamaleddin H. M. E. Tehrani, João Medeiros‐Silva, +19 more
46citations -
Adenosine receptors in GtoPdb v.2025.42025 IUPHAR/BPS Guide to Pharmacology CITE article Biochemistry, Genetics and Molecular Biology Adenosine and Purinergic Signaling Open access
Bertil B. Fredholm, U. Schwabe, Lauren Therese May, Christa Elisabeth Müller, Joel M Linden, Karl‐Norbert Klotz, +5 more
0citations -
Previously Published Phosphatase Probes have Limited Utility Due to their Unspecific Reactivity2024 ChemBioChem article Biochemistry, Genetics and Molecular Biology Protein Tyrosine Phosphatases Open access
Franciscus H. G. Ter Brake, Suzanne van Luttikhuizen, Tom van der Wel, Berend Gagestein, Bogdan I. Florea, Mario van der Stelt, +1 more
6citations -
Common characteristics of variants linked to autism spectrum disorder in the WAVE regulatory complex2025 Frontiers in Computational Neuroscience article Biochemistry, Genetics and Molecular Biology Genetics and Neurodevelopmental Disorders Open access
Song Xie, Ke Zuo, Silvia De Rubeis, Giorgio Bonollo, Giorgio Colombo, Paolo Ruggerone, +1 more
1citations -
Highly selective tyrosine kinase 2 inhibition with zasocitinib (TAK-279) improves outcomes in patients with active psoriatic arthritis: a randomised phase 2b study2025 Annals of the Rheumatic Diseases article Medicine Spondyloarthritis Studies and Treatments Open access
Alan Kivitz, Xenofon Baraliakos, Elena Tomaselli Muensterman, Arthur Kavanaugh, Désirée M F M van der Heijde, Piotr Adrian Klimiuk, +10 more
11citations -
Impact of cancer-associated mutations in CC chemokine receptor 2 on receptor function and antagonism2022 Biochemical Pharmacology article Biochemistry, Genetics and Molecular Biology Receptor Mechanisms and Signaling Open access
Lisa S. den Hollander, Olivier J. M. Béquignon, Xiangzi Wang, K. van Wezel, Jeremy D. Broekhuis, Marina Gorostiola González, +4 more
10citations -
Biomarker-Based Pharmacological Characterization of ENX-102, a Novel α2/3/5 Subtype-Selective GABAA Receptor Positive Allo-Steric Modulator: Translational Insights from Rodent and Human Studies
Paul Nettesheim, Krishna C. Vadodaria, Kimberly E. Vanover, Laura G. J. M. Borghans, Estibaliz Arce Cirauqui, Jordi Serrats, +5 more
0citations -
Inhibition of macrophage migration in zebrafish larvae demonstrates in vivo efficacy of human CCR2 inhibitors2020 Developmental & Comparative Immunology article Medicine Chemokine receptors and signaling Open access
Frida Sommer, Natalia V. Ortiz Zacarı́as, Laura H. Heitman, Annemarie H. Meijer
17citations