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Role of Conserved Tyrosine Lid Residues in the Activation of the M2 Muscarinic Acetylcholine Receptor2023 Molecular Pharmacology article Biochemistry, Genetics and Molecular Biology Receptor Mechanisms and Signaling Open access
Vi Pham, Maria Clazina Cornelia Habben Jansen, Geoff V. Thompson, Laura H. Heitman, Arthur Christopoulos, David M. Thal, +1 more
6citations -
Deciphering the allosteric control of androgen receptor DNA binding by its disordered N-terminal domain2025 Molecular and Cellular Endocrinology article Medicine Prostate Cancer Treatment and Research Open access
Laurens W.H.J. Heling, Adam P. Rofe, Andrea Alegre‐Martí, Vahid Sheikhhassani, Thomas Schmidt, Eva Estébanez‐Perpiñá, +2 more
2citations -
High-resolution cryo-EM structure of integrin αIIbβ3 bound to disease-causing maternal HPA-1a antibody that blocks integrin activation2026 bioRxiv (Cold Spring Harbor Laboratory) preprint Medicine Cell Adhesion Molecules Research Open access
José M. de Pereda, Wendy Stam, Marcos Gragera, Femke S. van der Meer, Francisco Javier Chichón, Eleftherios Zarkadas, +4 more
0citations -
Pilocarpine‐Induced Effects on Salivary Secretion as a Pharmacological Biomarker for Cholinergic Parasympathetic Activation2021 Clinical Pharmacology in Drug Development article Biochemistry, Genetics and Molecular Biology Receptor Mechanisms and Signaling
Nicoline Treijtel, Dorien Groenendaal‐van de Meent, Ingrid N. Michon, Cees Korstanje, John Meijer, Klaus Francke
5citations -
Allosteric control of Ubp6 and the proteasome via a bidirectional switch2021 bioRxiv (Cold Spring Harbor Laboratory) preprint Biochemistry, Genetics and Molecular Biology Ubiquitin and proteasome pathways Open access
Ka Ying Sharon Hung, Sven Klumpe, Markus R. Eisele, Suzanne Elsasser, Geng Tian, Shuangwu Sun, +13 more
5citations -
Allosteric control of Ubp6 and the proteasome via a bidirectional switch2022 Nature Communications article Biochemistry, Genetics and Molecular Biology Ubiquitin and proteasome pathways Open access
Ka Ying Sharon Hung, Sven Klumpe, Markus R. Eisele, Suzanne Elsasser, Geng Tian, Shuangwu Sun, +13 more
44citations -
Discovery of isoquinoline sulfonamides as allosteric gyrase inhibitors with activity against fluoroquinolone-resistant bacteria2024 Nature Chemistry article Biochemistry, Genetics and Molecular Biology Cancer therapeutics and mechanisms Open access
Alexander T. Bakker, Ioli Kotsogianni, Mariana Ávalos, Jeroen M. Punt, Bing Liu, Diana Piermarini, +13 more
29citations -
Structure of human spermine oxidase in complex with a highly selective allosteric inhibitor2022 Communications Biology article Biochemistry, Genetics and Molecular Biology Polyamine Metabolism and Applications Open access cited by 1 patent
Elsie Diaz, Suraj Adhikary, Armand W.J.W. Tepper, Daniel Riley, Rodrigo F. Ortiz‐Meoz, Daniel J. Krosky, +12 more
11citations -
Host defence peptide plectasin targets bacterial cell wall precursor lipid II by a calcium-sensitive supramolecular mechanism2024 Nature Microbiology article Immunology and Microbiology Antimicrobial Peptides and Activities Open access
Shehrazade Jekhmane, Maik G. N. Derks, Sourav Maity, Cornelis J. Slingerland, Kamaleddin H. M. E. Tehrani, João Medeiros‐Silva, +19 more
46citations -
Pharmacological Profiling of Antagonists for Cc Chemokine Receptor 5: Evidence for Allosterism, Biased Antagonism and Probe Dependence2025 SSRN Electronic Journal preprint Biochemistry, Genetics and Molecular Biology Receptor Mechanisms and Signaling Open access
Yao Yao, Gijs Stavast, Cas van der Horst, Natalia V. Ortiz Zacarı́as, Laura H. Heitman
0citations -
Adenosine receptors in GtoPdb v.2025.42025 IUPHAR/BPS Guide to Pharmacology CITE article Biochemistry, Genetics and Molecular Biology Adenosine and Purinergic Signaling Open access
Bertil B. Fredholm, U. Schwabe, Lauren Therese May, Christa Elisabeth Müller, Joel M Linden, Karl‐Norbert Klotz, +5 more
0citations -
Previously Published Phosphatase Probes have Limited Utility Due to their Unspecific Reactivity2024 ChemBioChem article Biochemistry, Genetics and Molecular Biology Protein Tyrosine Phosphatases Open access
Franciscus H. G. Ter Brake, Suzanne van Luttikhuizen, Tom van der Wel, Berend Gagestein, Bogdan I. Florea, Mario van der Stelt, +1 more
6citations -
Common characteristics of variants linked to autism spectrum disorder in the WAVE regulatory complex2025 Frontiers in Computational Neuroscience article Biochemistry, Genetics and Molecular Biology Genetics and Neurodevelopmental Disorders Open access
Song Xie, Ke Zuo, Silvia De Rubeis, Giorgio Bonollo, Giorgio Colombo, Paolo Ruggerone, +1 more
1citations -
Structures of Arabidopsis thaliana MDL Proteins and Synergistic Effects with the Cytokine MIF on Human Receptors2023 bioRxiv (Cold Spring Harbor Laboratory) preprint Immunology and Microbiology Macrophage Migration Inhibitory Factor Open access
Lukas Spiller, R. Manjula, Franz Leissing, J. Basquin, Priscila Bourilhon, Dzmitry Sinitski, +8 more
0citations