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Methyl substituted β –lactam framework based antibiotics and β -lactamase inhibitors: Proof of concept by computations2024 bioRxiv (Cold Spring Harbor Laboratory) preprint Chemistry Synthesis of β-Lactam Compounds Open access
Vaishali Thakkur, Chandan Kumar Das, Shivani Verma, Suman Saha, Nisanth N. Nair
0citations -
High-throughput quantification of ochronotic pigment formation in Escherichia coli to evaluate the potency of human 4-hydroxyphenylpyruvate dioxygenase inhibitors in multi-well format2020 MethodsX article Biochemistry, Genetics and Molecular Biology Metabolism and Genetic Disorders Open access
Jessie Neuckermans, Sien Lequeue, Alan Mertens, Steven Branson, Ulrich Schwaneberg, Joery De Kock
2citations -
Structure–Activity Relationship Studies of Pyrimidine-4-Carboxamides as Inhibitors of N -Acylphosphatidylethanolamine Phospholipase D2020 Journal of Medicinal Chemistry article Medicine Cannabis and Cannabinoid Research Open access cited by 1 patent
Elliot D. Mock, Ioli Kotsogianni, Wouter P. F. Driever, Carmen S. Fonseca, Jelle M. Vooijs, Hans den Dulk, +2 more
9citations -
Association of Polymorphic Cytochrome P450 Enzyme Pathways with Falls in Multimedicated Older Adults2024 Journal of the American Medical Directors Association article Pharmacology, Toxicology and Pharmaceutics Pharmacogenetics and Drug Metabolism Open access
Katja Susanne Just, Laura M. Pott, Catharina Scholl, Michael Steffens, Michael Dieter Denkinger, Dietrich Rothenbacher, +2 more
4citations -
Immobilized-enzyme reactors integrated into analytical platforms: Recent advances and challenges2021 TrAC Trends in Analytical Chemistry article Biochemistry, Genetics and Molecular Biology Enzyme Catalysis and Immobilization Open access
Bert Wouters, Sinéad Currivan, Noor Abdulhussain, Thomas Hankemeier, Peter J. Schoenmakers
61citations -
Development of Potent and Selective Monoacylglycerol Lipase Inhibitors. SARs, Structural Analysis, and Biological Characterization2024 Journal of Medicinal Chemistry article Medicine Cholinesterase and Neurodegenerative Diseases Open access
Stefania Butini, Uwe Grether, Kwang‐Mook Jung, Alessia Ligresti, Marco Allarà, Annemarieke G. J. Postmus, +18 more
8citations -
Discovery and Optimization of a Novel Series of Pyrazolopyrimidines as Spermine Oxidase Inhibitors2025 Journal of Medicinal Chemistry article Biochemistry, Genetics and Molecular Biology Polyamine Metabolism and Applications
Josep Llaveria, Suraj Adhikary, Christophe Buyck, Santiago Cañellas, Jose Maria Cid, Ben Danna, +14 more
0citations -
From dual norepinephrine–dopamine reuptake inhibition to selective dopamine reuptake inhibitors: a case of aromatically substituted N ,2-cyclopentylamines2026 RSC Medicinal Chemistry article Neuroscience Neurotransmitter Receptor Influence on Behavior Open access
Majlen A. Dilweg, Willem Jespers, Ameya Sanjay Kasture, Rongfang Liu, Tamara A. M. Mocking, Jelle G Van Der Ploeg, +7 more
0citations -
Effects of Angiotensin-Converting Enzyme Inhibition on the Recurrence and Internal Structure of Chronic Subdural Hematomas2024 Journal of Clinical Medicine article Medicine Neurosurgical Procedures and Complications Open access
Michael Veldeman, Hani Ridwan, Mohamed Alzaiyani, Rastislav Pjontek, Benedikt Kremer, Anke Höllig, +2 more
6citations -
Multiplexed Gel-based ABPP Strategy for Target-agnostic Serine Hydrolase Inhibitor Screening2026 CHIMIA International Journal for Chemistry article Chemistry Click Chemistry and Applications Open access
Franciscus H. G. Ter Brake, Patrick Rehorst, Machiel W. Henst, Mario van der Stelt, Antonius P. A. Janssen
1citations -
Hypothesis-Driven, Structure-Based Design in Photopharmacology: The Case of eDHFR Inhibitors2022 Journal of Medicinal Chemistry article Materials Science Photochromic and Fluorescence Chemistry Open access
Piermichele Kobauri, Nicole Stéphanie Galenkamp, Albert Marten Schulte, Jisk de Vries, Nadja A. Simeth, Giovanni Maglia, +4 more
27citations -
Macrocyclic peptides as allosteric inhibitors of nicotinamide N -methyltransferase (NNMT)2021 RSC Chemical Biology article Biochemistry, Genetics and Molecular Biology Biochemical and Molecular Research Open access cited by 3 patents
Matthijs J. van Haren, Yurui Zhang, Vito Thijssen, Ned P. Buijs, Yongzhi Gao, Łukasz Mateuszuk, +8 more
62citations -
High‐Throughput Synthesis and Screening of a Cyanimide Library Identifies Selective Inhibitors of ISG15‐Specific Protease mUSP182025 Angewandte Chemie International Edition article Biochemistry, Genetics and Molecular Biology Chemical Synthesis and Analysis Open access
Raymond Kooij, Vito Pol, Bjorn R. van Doodewaerd, Ayşegül Sapmaz, Marta Campos Alonso, Günter Fritz, +2 more
7citations -
High-Throughput Synthesis and Screening of a Cyanimide Library Identifies Selective Inhibitors of ISG15-specific Protease USP182025 bioRxiv (Cold Spring Harbor Laboratory) preprint Biochemistry, Genetics and Molecular Biology Chemical Synthesis and Analysis Open access
Raymond Kooij, Vito Pol, Bjorn R. van Doodewaerd, Ayşegül Sapmaz, Günter Fritz, Klaus‐Peter Knobeloch, +1 more
2citations -
High‐Throughput Synthesis and Screening of a Cyanimide Library Identifies Selective Inhibitors of ISG15‐Specific Protease mUSP182025 Angewandte Chemie article Biochemistry, Genetics and Molecular Biology Chemical Synthesis and Analysis Open access
Raymond Kooij, Vito Pol, Bjorn R. van Doodewaerd, Ayşegül Sapmaz, Marta Campos Alonso, Günter Fritz, +2 more
0citations -
Aminocarboxylic acids related to aspergillomarasmine A (AMA) and ethylenediamine- N , N ′-disuccinic acid (EDDS) are strong zinc-binders and inhibitors of the metallo-beta-lactamase NDM-1
Kamaleddin H. M. E. Tehrani, Haigen Fu, Nora C. Brüchle, Vida Mashayekhi, Alejandro Prats Luján, Matthijs J. van Haren, +2 more
22citations