Papers matching “P-glycoprotein inhibitors” 18
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Measurement of cyclosporin induced changes in P-glycoprotein function at the human blood-brain barrier using [18F]MC225 and PET2025 European Journal of Nuclear Medicine and Molecular Imaging article Medicine Drug Transport and Resistance Mechanisms Open access
Pascalle Mossel, Giordana Salvi de Souza, Antoon T. M. Willemsen, Gilles N. Stormezand, Nicola Antonio Colabufo, Jun Toyohara, +5 more
5citations -
Do P-glycoprotein-mediated drug-drug interactions at the blood-brain barrier impact morphine brain distribution?2025 Journal of Pharmacokinetics and Pharmacodynamics article Medicine Drug Transport and Resistance Mechanisms Open access
Berfin Gülave, Ariel Lesmana, Elizabeth C. M. de Lange, J. G. Coen van Hasselt
4citations -
Mapping cardiac drug transport: In vitro assessment of cardiac P-glycoprotein function with [18F]MC225 by using µ-engineered heart tissues2025 European Heart Journal Open article Medicine Drug Transport and Resistance Mechanisms Open access
Wanling Liu, Maureen Dannenberg, Pascalle Mossel, Zeyu Cai, Ines Farinha Antunes, Jürgen W. A. Sijbesma, +7 more
1citations -
A New ABCB1 Inhibitor Enhances the Anticancer Effect of Doxorubicin in Both In Vitro and In Vivo Models of NSCLC2023 International Journal of Molecular Sciences article Medicine Drug Transport and Resistance Mechanisms Open access
Maria Pia Adorni, Maricla Galetti, Silvia La Monica, Matteo Incerti, Alessandro Ruffoni, Lisa Elviri, +6 more
16citations -
The human proton pump inhibitors inhibit Mycobacterium tuberculosis rifampicin efflux and macrophage-induced rifampicin tolerance2023 Proceedings of the National Academy of Sciences article Medicine Tuberculosis Research and Epidemiology Open access
M. Alexandra Lake, Kristin N. Adams, Feilin Nie, Elaine Fowler, Amit Kumar Verma, Silvia Dei, +6 more
33citations -
ABCB1 overexpression through locus amplification represents an actionable target to combat paclitaxel resistance in pancreatic cancer cells2023 bioRxiv (Cold Spring Harbor Laboratory) preprint Medicine Drug Transport and Resistance Mechanisms Open access
Cecilia Bergonzini, Alessandro Gregori, Tessa M. S. Hagens, Vera E. van der Noord, Bob van de Water, Annelien J.M. Zweemer, +9 more
1citations -
Physiologically‐based pharmacokinetic modeling of quinidine to establish a CYP3A4 , P‐gp, and CYP2D6 drug–drug–gene interaction network2023 CPT Pharmacometrics & Systems Pharmacology article Pharmacology, Toxicology and Pharmaceutics Pharmacogenetics and Drug Metabolism Open access
Denise Feick, Simeon Rüdesheim, Fatima Zahra Marok, Dominik Selzer, Helena Leonie Hanae Loer, Donato Teutonico, +6 more
12citations -
Editorial: Innovations in pharmacogenomics: embracing diversity and clinical application2026 Frontiers in Pharmacology editorial Pharmacology, Toxicology and Pharmaceutics Pharmacogenetics and Drug Metabolism Open access
Maaike van der Lee, Sarah Cargnin, Elena Peruzzi, Claudia Pisanu, Rossana Roncato
0citations -
A Comprehensive CYP2D6 Drug–Drug–Gene Interaction Network for Application in Precision Dosing and Drug Development2025 Clinical Pharmacology & Therapeutics article Pharmacology, Toxicology and Pharmaceutics Pharmacogenetics and Drug Metabolism Open access
Simeon Rüdesheim, Helena Leonie Hanae Loer, Denise Feick, Fatima Zahra Marok, Laura Maria Fuhr, Dominik Selzer, +9 more
15citations -
Multi-parameter optimization: Development of a morpholin-3-one derivative with an improved kinetic profile for imaging monoacylglycerol lipase in the brain2022 European Journal of Medicinal Chemistry article Medicine Cannabis and Cannabinoid Research Open access
Yingfang He, Uwe Grether, Marco F. Taddio, Carla Meier, Claudia Keller, Martin R. Edelmann, +14 more
14citations -
ABCB1 overexpression through locus amplification represents an actionable target to combat paclitaxel resistance in pancreatic cancer cells2024 Journal of Experimental & Clinical Cancer Research article Medicine Drug Transport and Resistance Mechanisms Open access
Cecilia Bergonzini, Alessandro Gregori, Tessa M. S. Hagens, Vera E. van der Noord, Bob van de Water, Annelien J.M. Zweemer, +10 more
38citations -
685P Genome-wide association meta-analysis identifies novel variants that correlate with efficacy outcomes in sunitinib-treated patients with metastatic renal cell carcinoma
Meta H.M. Diekstra, Jesse Joachim Swen, L. van der Zanden, Epic Boven, Ron H.J. Mathijssen, Arna Óskarsdóttir, +13 more
0citations -
Extrahepatic metabolism of ibrutinib2020 Investigational New Drugs article Pharmacology, Toxicology and Pharmaceutics Pharmacogenetics and Drug Metabolism Open access
Johannes J.M. Rood, Amer Jamalpoor, Stéphanie van Hoppe, Matthijs J. van Haren, Roeland E. Wasmann, Manoe Jacoba Janssen, +4 more
28citations -
Should we abandon therapeutic drug monitoring of tacrolimus in whole blood and move to intracellular concentration measurements?2023 British Journal of Clinical Pharmacology article Medicine Renal Transplantation Outcomes and Treatments Open access
Suwasin Udomkarnjananun, Thanee Eiamsitrakoon, Brenda C. M. de Winter, Teun van Gelder, Dennis Alexander Hesselink
19citations
18 results