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The sodium‐glucose co‐transporter‐2 inhibitor ertugliflozin modifies the signature of cardiac substrate metabolism and reduces cardiac mTOR signalling, endoplasmic reticulum stress and apoptosis
Julia Moellmann, Pascal A. Mann, Ben Arpad Kappel, Florian Kahles, Barbara M. Klinkhammer, Peter Boor, +5 more
52citations -
Navigating Solute Carrier Transporters—A Comprehensive Review of Functionalized Small Molecule Probes for Target Identification and Characterization2025 Medicinal Research Reviews review Medicine Drug Transport and Resistance Mechanisms Open access
Majlen A. Dilweg, Tracie Widjaja, Adriaan P. IJzerman, Daan van der Es
2citations -
MPP+-Induced Changes in Cellular Impedance as a Measure for Organic Cation Transporter (SLC22A1-3) Activity and Inhibition2022 International Journal of Molecular Sciences article Medicine Drug Transport and Resistance Mechanisms Open access
Tamara A. M. Mocking, Hubert J. Sijben, Yimé Vermeulen, Adriaan P. IJzerman, Laura H. Heitman
5citations -
Identification and characterization of nanobodies specific for the human ubiquitin–like ISG15 protein2025 Journal of Biological Chemistry article Medicine Monoclonal and Polyclonal Antibodies Research Open access cited by 1 patent
Prachi Dabhade, Charlotte Wijne, William McKibben, Simeon D. Draganov, Hedib Alkoumi H Alrawili, Zhen-Yu Jim Sun, +8 more
3citations -
Mapping cardiac drug transport: In vitro assessment of cardiac P-glycoprotein function with [18F]MC225 by using µ-engineered heart tissues2025 European Heart Journal Open article Medicine Drug Transport and Resistance Mechanisms Open access
Wanling Liu, Maureen Dannenberg, Pascalle Mossel, Zeyu Cai, Ines Farinha Antunes, Jürgen W. A. Sijbesma, +7 more
1citations
16 results