September 27, 2007 article Fluorine in Pharmaceuticals: Looking Beyond Intuition Science DOI: 10.1126/science.1131943 OpenAlex Authors 0 Author list not loaded yet. Cited by 24 stored of 6,642 Search Sort Most cited Newest Oldest Patent citations Title Any typearticle review book-chapter conference-paper preprint dissertation book dataset other Any fieldAgricultural and Biological Sciences Arts and Humanities Biochemistry, Genetics and Molecular Biology Business, Management and Accounting Chemical Engineering Chemistry Computer Science Decision Sciences Dentistry Earth and Planetary Sciences Economics, Econometrics and Finance Energy Engineering Environmental Science Health Professions Immunology and Microbiology Materials Science Mathematics Medicine Neuroscience Nursing Pharmacology, Toxicology and Pharmaceutics Physics and Astronomy Psychology Social Sciences Veterinary Open access Charting New Territory: Systematic Evaluation of the Drug Potential of N -Trifluoromethyl Amides, Ureas & Carbamates 2026 Journal of Medicinal Chemistry article Pharmacology, Toxicology and Pharmaceutics Fluorine in Organic Chemistry Open access 2 citations Access to N ‐Monofluoromethylated (Thio)Carbamates, Formamides, Alkynamides, and Related Derivatives 2025 Angewandte Chemie International Edition article Pharmacology, Toxicology and Pharmaceutics Fluorine in Organic Chemistry Open access 11 citations Access to N ‐Monofluoromethylated (Thio)Carbamates, Formamides, Alkynamides, and Related Derivatives 2025 Angewandte Chemie article Pharmacology, Toxicology and Pharmaceutics Fluorine in Organic Chemistry Open access 2 citations Desulfurizative Fluorination of N ‐CF 3 Thioformamides for the Efficient Synthesis of N (CF 3 )(CF 2 H) Amines with Enhanced Stability 2025 Angewandte Chemie International Edition article Pharmacology, Toxicology and Pharmaceutics Fluorine in Organic Chemistry Open access 5 citations Desulfurizative Fluorination of N ‐CF 3 Thioformamides for the Efficient Synthesis of N (CF 3 )(CF 2 H) Amines with Enhanced Stability 2025 Angewandte Chemie article Pharmacology, Toxicology and Pharmaceutics Fluorine in Organic Chemistry Open access 1 citations A Photo- and Electrochemistry-Triggered Redox-Neutral Cyclization Strategy to Access Cyclic N -CF 3 Amides 2025 Organic Letters article Chemistry Radical Photochemical Reactions 6 citations Mechanochemical difluoromethylations of ketones 2024 Beilstein Journal of Organic Chemistry article Pharmacology, Toxicology and Pharmaceutics Fluorine in Organic Chemistry Open access 7 citations Mechanistic Insights on the Challenging Trifluoromethylation of Ni(II) 2024 ACS Catalysis article Pharmacology, Toxicology and Pharmaceutics Fluorine in Organic Chemistry 3 citations Access to N -Difluoromethyl Amides, (Thio)Carbamates, Ureas, and Formamides 2024 Journal of the American Chemical Society article Pharmacology, Toxicology and Pharmaceutics Fluorine in Organic Chemistry Open access cited by 1 patent 47 citations Homologation Reactions for the Synthesis of Fluorinated Molecules 2023 other Pharmacology, Toxicology and Pharmaceutics Fluorine in Organic Chemistry Open access 0 citations Access to N −CF 3 Formamides by Reduction of N −CF 3 Carbamoyl Fluorides 2022 Angewandte Chemie International Edition article Pharmacology, Toxicology and Pharmaceutics Fluorine in Organic Chemistry Open access 47 citations Access to N−CF3 Formamides by Reduction of N−CF3 Carbamoyl Fluorides 2022 Angewandte Chemie article Pharmacology, Toxicology and Pharmaceutics Fluorine in Organic Chemistry Open access 4 citations N‐CF3 Imidazolidin‐2‐one Derivatives via Photocatalytic and Silver‐Catalyzed Cyclizations 2022 Chemistry - 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