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• ▲ Herman S. Overkleeft

  Leiden University · Scripps Research Institute Chemistry
  29k

  citations

  84

  h-index

  163

  Aachen papers
• ▲ Gijsbert A. van der Marel

  Leiden University Chemistry
  14.6k

  citations

  60

  h-index

  74

  Aachen papers
• ▲ Jeroen D. C. Codée

  Leiden University · Scripps Research Institute Chemistry
  10.9k

  citations

  55

  h-index

  165

  Aachen papers
• ▲ Gijs A. van der MAREL

  Leiden University Chemistry
  10.5k

  citations

  53

  h-index

  12

  Aachen papers
• ▲ Dmitri V. Filippov

  Leiden University Biochemistry, Genetics and Molecular Biology
  8.54k

  citations

  47

  h-index

  86

  Aachen papers
• ▲ Bogdan I. Florea

  Leiden University · Netherlands Proteomics Centre Biochemistry, Genetics and Molecular Biology
  7.56k

  citations

  50

  h-index

  48

  Aachen papers
• ▲ Hans van den Elst

  Leiden University · Leiden University Medical Center Biochemistry, Genetics and Molecular Biology
  3.8k

  citations

  29

  h-index

  8

  Aachen papers
• ▲ Fabrizio Chiodo

  Institute for Biomedical Research and Innovation · Istituto di Chimica Biomolecolare Biochemistry, Genetics and Molecular Biology
  2.35k

  citations

  28

  h-index

  4

  Aachen papers
• ▲ Nico J. Meeuwenoord

  Leiden University Biochemistry, Genetics and Molecular Biology
  2.18k

  citations

  28

  h-index

  18

  Aachen papers
• ▲ Marta Artola

  Leiden University · Leiden University Medical Center Chemistry
  1.95k

  citations

  26

  h-index

  39

  Aachen papers
• ▲ Jan Dijk

  Leiden University Biochemistry, Genetics and Molecular Biology
  1.87k

  citations

  22

  h-index

  1

  Aachen papers
• ▲ Zachary Armstrong

  Leiden University Chemistry
  826

  citations

  16

  h-index

  22

  Aachen papers
• ▲ Florian Küllmer

  Leiden University · Leiden University Medical Center Biochemistry, Genetics and Molecular Biology
  450

  citations

  7

  h-index

  4

  Aachen papers
• ▲ Valentina Borlandelli

  Leiden University · University of Basel Biochemistry, Genetics and Molecular Biology
  441

  citations

  8

  h-index

  11

  Aachen papers
• ▲ Jim Voorneveld

  Leiden University Biochemistry, Genetics and Molecular Biology
  359

  citations

  10

  h-index

  13

  Aachen papers
• ▲ Niels R. M. Reintjens

  University of Groningen Chemistry
  272

  citations

  9

  h-index

  4

  Aachen papers
• ▲ Sven Wijngaarden

  Leiden University · Leiden University Medical Center Biochemistry, Genetics and Molecular Biology
  245

  citations

  9

  h-index

  15

  Aachen papers
• ▲ Ana R. de Jong

  Leiden University Chemistry
  230

  citations

  5

  h-index

  1

  Aachen papers
• ▲ Hugo Minnee

  Leiden University Chemistry
  104

  citations

  6

  h-index

  9

  Aachen papers
• ▲ Jacopo Enotarpi

  Leiden University Chemistry
  96

  citations

  5

  h-index

  9

  Aachen papers
• ▲ Marjolein M. E. Isendoorn

  Leiden University Immunology and Microbiology
  84

  citations

  3

  h-index

  9

  Aachen papers
• ▲ Evert Peterse

  Amsterdam UMC Location Vrije Universiteit Amsterdam Immunology and Microbiology
  78

  citations

  3

  h-index

  4

  Aachen papers
• ▲ Lars C. P. Binkhorst

  Biochemistry, Genetics and Molecular Biology
  18

  citations

  3

  h-index

  1

  Aachen papers
• ▲ Hayley Chung

  Leiden University Chemistry
  12

  citations

  1

  h-index

  1

  Aachen papers
• ▲ Femke L. A. M. van der Heijden

  Leiden University Chemistry
  8

  citations

  2

  h-index

  5

  Aachen papers
• ▲ Vincent V. F. Verhoeks

  Leiden University Medicine
  7

  citations

  1

  h-index

  3

  Aachen papers
• ▲ Moescha Hoopman

  Leiden University Chemistry
  6

  citations

  1

  h-index

  2

  Aachen papers

27 results

• Discovery of a NAPE-PLD inhibitor that modulates emotional behavior in mice

  2020 Nature Chemical Biology article Medicine Cannabis and Cannabinoid Research Open access

  99

  citations
• Unbiased Identification of the Liposome Protein Corona using Photoaffinity-based Chemoproteomics

  2020 ACS Central Science article Materials Science Nanoparticle-Based Drug Delivery Open access cited by 1 patent

  72

  citations
• Chemoenzymatic and Synthetic Approaches To Investigate Aspartate- and Glutamate-ADP-Ribosylation

  2023 Journal of the American Chemical Society article Biochemistry, Genetics and Molecular Biology Chemical Synthesis and Analysis Open access cited by 1 patent

  53

  citations
• Self-Adjuvanting Cancer Vaccines from Conjugation-Ready Lipid A Analogues and Synthetic Long Peptides

  2020 Journal of Medicinal Chemistry article Immunology and Microbiology Immunotherapy and Immune Responses Open access cited by 7 patents

  37

  citations
• Arginine ADP-Ribosylation: Chemical Synthesis of Post-Translationally Modified Ubiquitin Proteins

  2022 Journal of the American Chemical Society article Biochemistry, Genetics and Molecular Biology Chemical Synthesis and Analysis Open access

  29

  citations
• Synthetic Oligomers Mimicking Capsular Polysaccharide Diheteroglycan are Potential Vaccine Candidates against Encapsulated Enterococcal Infections

  2020 ACS Infectious Diseases article Chemistry Carbohydrate Chemistry and Synthesis Open access cited by 3 patents

  28

  citations
• Comparative Photoaffinity Profiling of Omega-3 Signaling Lipid Probes Reveals Prostaglandin Reductase 1 as a Metabolic Hub in Human Macrophages

  2022 Journal of the American Chemical Society article Nursing Fatty Acid Research and Health Open access

  24

  citations
• Mimetics of ADP-Ribosylated Histidine through Copper(I)-Catalyzed Click Chemistry

  2022 Organic Letters article Chemistry Click Chemistry and Applications Open access cited by 1 patent

  16

  citations
• Legionella metaeffector MavL reverses ubiquitin ADP-ribosylation via a conserved arginine-specific macrodomain

  2024 Nature Communications article Biochemistry, Genetics and Molecular Biology Ubiquitin and proteasome pathways Open access

  16

  citations
• Chemical Proteomics Reveals Off-Targets of the Anandamide Reuptake Inhibitor WOBE437

  2022 ACS Chemical Biology article Medicine Cannabis and Cannabinoid Research Open access

  13

  citations
• Four of a Kind: A Complete Collection of ADP-Ribosylated Histidine Isosteres Using Cu(I)- and Ru(II)-Catalyzed Click Chemistry

  2023 The Journal of Organic Chemistry article Chemistry Click Chemistry and Applications Open access

  12

  citations
• Solid‐Phase Synthesis and Biological Evaluation of Peptides ADP‐Ribosylated at Histidine

  2023 Angewandte Chemie International Edition article Biochemistry, Genetics and Molecular Biology Chemical Synthesis and Analysis Open access

  11

  citations
• Lipid A analog CRX-527 conjugated to synthetic peptides enhances vaccination efficacy and tumor control

  2022 npj Vaccines article Immunology and Microbiology Immunotherapy and Immune Responses Open access

  10

  citations
• CellEKT: A Robust Chemical Proteomics Workflow to Profile Cellular Target Engagement of Kinase Inhibitors

  2025 Molecular & Cellular Proteomics article Chemistry Advanced Proteomics Techniques and Applications Open access

  8

  citations
• 4‐O‐Substituted Glucuronic Cyclophellitols are Selective Mechanism‐Based Heparanase Inhibitors

  2022 ChemMedChem article Chemistry Carbohydrate Chemistry and Synthesis Open access

  8

  citations
• β- l - Arabino furano-cyclitol Aziridines Are Covalent Broad-Spectrum Inhibitors and Activity-Based Probes for Retaining β- l -Arabinofuranosidases

  2023 ACS Chemical Biology article Chemistry Carbohydrate Chemistry and Synthesis Open access

  8

  citations
• Evolutionary and molecular basis of ADP-ribosylation reversal by zinc-dependent macrodomains

  2024 Journal of Biological Chemistry article Biochemistry, Genetics and Molecular Biology Biochemical and Molecular Research Open access

  8

  citations
• Mycobacterial Phenolic Glycolipid Triggers ATP-Mediated Neuronal P2X3 Signaling and Cough

  2025 bioRxiv (Cold Spring Harbor Laboratory) preprint Medicine Respiratory and Cough-Related Research Open access

  6

  citations
• Chemical Synthesis of Native ADP-Ribosylated Oligonucleotides Enables Analysis of DNA ADP-Ribosylation Hydrolase Specificity

  2026 Journal of the American Chemical Society article Biochemistry, Genetics and Molecular Biology DNA and Nucleic Acid Chemistry Open access

  4

  citations
• 6-O-alkyl 4-methylumbelliferyl-β-D-glucosides as selective substrates for GBA1 in the discovery of glycosylated sterols

  2024 Journal of Lipid Research article Medicine Lysosomal Storage Disorders Research Open access

  2

  citations