Synthesis of 3-amino-substituted benzothiadiazine oxides by a palladium-catalysed cascade reaction

Green Chemistry, vol. 25, pp. 3021–3026

Abstract

By using a very low catalyst loading, a wide range of cyclic sulfoximine derivatives, that represent common cores of bioactive products, can be prepared in good to excellent yields at room temperature in a short period of time.

Authors 6

1. Renè Hommelsheim Aachen Institute of Organic Chemistry

   RWTH Aachen University

   Affiliation as printed

   Institute of Organic Chemistry, RWTH Aachen University, Landoltweg 1, D-52074 Aachen, Germany

2. Sandra Bausch Aachen Institute of Organic Chemistry

   RWTH Aachen University

   Affiliation as printed

   Institute of Organic Chemistry, RWTH Aachen University, Landoltweg 1, D-52074 Aachen, Germany

3. Robin van Nahl Aachen Institute of Organic Chemistry

   RWTH Aachen University

   Affiliation as printed

   Institute of Organic Chemistry, RWTH Aachen University, Landoltweg 1, D-52074 Aachen, Germany

4. Jas S. Ward

   University of Jyväskylä

   Affiliation as printed

   University of Jyvaskyla, Department of Chemistry, FI-40014 Jyväskylä, Finland

5. Kari T. Rissanen

   University of Jyväskylä

   Affiliation as printed

   University of Jyvaskyla, Department of Chemistry, FI-40014 Jyväskylä, Finland

6. Carsten Bolm corresponding Aachen Institute of Organic Chemistry

   RWTH Aachen University

   Affiliation as printed

   Institute of Organic Chemistry, RWTH Aachen University, Landoltweg 1, D-52074 Aachen, Germany